2661-2673
| 2-Carbomethoxy-3-aryl-8-oxabicyclo[3.2.1]octanes: Potent Non-Nitrogen Inhibitors of Monoamine Transporters
Peter C. Meltzer,
Anna Y. Liang,
Paul Blundell,
Mario D. Gonzalez,
Zhengming Chen,
Clifford George, and
Bertha K. Madras
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2674-2687
| N-Arylpiperazinyl-N'-propylamino Derivatives of Heteroaryl Amides as Functional Uroselective  1-Adrenoceptor Antagonists
Todd R. Elworthy,
Anthony P. D. W. Ford,
Gary W. Bantle,
David J. Morgans, Jr.,
Rachel S. Ozer,
Wylie S. Palmer,
David B. Repke,
Magarita Romero,
Leticia Sandoval,
Eric B. Sjogren,
Francisco X. Talamás,
Alfredo Vazquez,
Helen Wu,
Nicolas F. Arredondo,
David R. Blue, Jr.,
Andrea DeSousa,
Lisa M. Gross,
M. Shannon Kava,
John D. Lesnick,
Rachel L. Vimont,
Timothy J. Williams,
Quan-Ming Zhu,
Jürg R. Pfister, and
David E. Clarke
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2688-2693
| Chromeno[3,4-c]pyridin-5-ones: Selective Human Dopamine D4 Receptor Antagonists as Potential Antipsychotic Agents
Paul C. Unangst,
Thomas Capiris,
David T. Connor,
Thomas G. Heffner,
Robert G. MacKenzie,
Steven R. Miller,
Thomas A. Pugsley, and
Lawrence D. Wise
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2694-2705
| Synthesis, Biological Evaluation, and Structure-Activity Relationships of 3-Acylindole-2-carboxylic Acids as Inhibitors of the Cytosolic Phospholipase A2
Matthias Lehr
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2706-2725
| Optimization of 3-(1H-Indazol-3-ylmethyl)-1,5-benzodiazepines as Potent, Orally Active CCK-A Agonists
Brad R. Henke,
Christopher J. Aquino,
Larry S. Birkemo,
Dallas K. Croom,
Robert W. Dougherty, Jr.,
Gregory N. Ervin,
Mary K. Grizzle,
Gavin C. Hirst,
Michael K. James,
Michael F. Johnson,
Kennedy L. Queen,
Ronald G. Sherrill,
Elizabeth E. Sugg,
Edward M. Suh,
Jerzy W. Szewczyk,
Rayomand J. Unwalla,
Jeff Yingling, and
Timothy M. Willson
[Full Article -
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2726-2732
| Synthesis and Antimalarial Effects of Phenothiazine Inhibitors of a Plasmodium falciparum Cysteine Protease
José N. Domínguez,
Simón López,
Jaime Charris,
Lúcido Iarruso,
Gricela Lobo,
Andrey Semenov,
Jed E. Olson, and
Philip J. Rosenthal
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2733-2739
| Synthesis and Opioid Activity of [D-Pro10]Dynorphin A-(1-11) Analogues with N-Terminal Alkyl Substitution
Heekyung Choi,
Thomas F. Murray,
Gary E. DeLander,
William K. Schmidt, and
Jane V. Aldrich
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2740-2749
|  -Methylation of the Phe7 and Trp9 Melanotropin Side Chain Pharmacophores Affects Ligand-Receptor Interactions and Prolonged Biological Activity
Carrie Haskell-Luevano,
Kate Toth,
Lakmal Boteju,
Constatin Job,
Ana Maria de L. Castrucci,
Mac E. Hadley, and
Victor J. Hruby
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2750-2754
| Synthesis and Anti-Hepatitis B Virus Activity of 9-(2-Deoxy-2-fluoro--L-arabinofuranosyl)purine Nucleosides
Tianwei Ma,
Ju-Sheng Lin,
M. Gary Newton,
Yung-Chi Cheng, and
Chung K. Chu
[Full Article -
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2755-2761
| 6A-O-[(4-Biphenylyl)acetyl]--, --, and - -cyclodextrins and 6A-Deoxy-6A-[[(4-biphenylyl)acetyl]amino]--, --, and --cyclodextrins: Potential Prodrugs for Colon-Specific Delivery
Kaneto Uekama,
Kunihiro Minami, and
Fumitoshi Hirayama
[Full Article -
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2762-2769
| Novel Agonists of 5HT2C Receptors. Synthesis and Biological Evaluation of Substituted 2-(Indol-1-yl)-1-methylethylamines and 2-(Indeno[1,2-b]pyrrol-1-yl)-1-methylethylamines. Improved Therapeutics for Obsessive Compulsive Disorder
Michael Bös,
François Jenck,
James R. Martin,
Jean-Luc Moreau,
Andrew J. Sleight,
Jürgen Wichmann, and
Ulrich Widmer
[Full Article -
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2770-2779
| Synthesis, Photophysical Properties, in Vivo Photosensitizing Efficacy, and Human Serum Albumin Binding Properties of Some Novel Bacteriochlorins
Ravindra K. Pandey,
Scott Constantine,
Takaaki Tsuchida,
Gang Zheng,
Craig J. Medforth,
Mohamed Aoudia,
Andrei N. Kozyrev,
Michael A. J. Rodgers,
Harubumi Kato,
Kevin M. Smith, and
Thomas J. Dougherty
[Full Article -
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2780-2787
| Antipsoriatic Anthrones with Modulated Redox Properties. 4. Synthesis and Biological Activity of Novel 9,10-Dihydro-1,8-dihydroxy-9-oxo-2- anthracenecarboxylic and -hydroxamic Acids
Klaus Müller and
Helge Prinz
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2788-2792
| Immunologically Specific Activation of a Cephalosporin Derivative of Mitomycin C by Monoclonal Antibody -Lactamase Conjugates
Vivekananda M. Vrudhula,
Håkan P. Svensson, and
Peter D. Senter
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